山东大学教师主页康东伟 Paper Publications Home

康东伟

Professor
Supervisor of Master's Candidates

Gender:Male
Education Level:With Certificate of Graduation for Doctorate Study
Degree:Doctoral Degree in Medicine
Status:Employed
School/Department:药学院
Date of Employment:2020-10-22
College: Cheeloo College of Medicine
Discipline:Medicinal Chemistry

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Current position: Home >> Scientific Research >> Paper Publications

Paper Publications

2021-09
[1] 黄伯世. Structure-Based Design and Discovery of Pyridyl-Bearing Fused Bicyclic HIV-1 Inhibitors: Synthesis, Biological Characterization, and Molecular Modeling Studies. Journal of Medicianal Chemistry, 64, 13604-13621, 2021.
2018-05
[2] 黄伯世. First discovery of a potential carbonate prodrug of NNRTI drug candidate RDEA427 with submicromolar inhibitory activity against HIV-1 K103N/Y181C double mutant strain. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 28, 1348, 2018.
2020-12
[3] 郑义. Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) membrane (M) protein inhibits type I and III interferon production by targeting RIG-I/MDA-5 signaling. SIGNAL TRANSDUCTION AND TARGETED THERAPY, 5, 2020.
2019-08
[4] 刘新泳. Recent applications of click chemistry in drug discovery. Expert Opin Drug Discov, 2019.
2019-05
[5] 刘新泳. Overview of Recent Strategic Advances in Medicinal Chemistry. J Med Chem, 2019.
2018-12
[6] 刘新泳. Development of a practical synthesis of etravirine via a microwave-promoted amination. chemistry central Journal, 2018.
2021-01
[7] 黄伯世. Design, synthesis, and biological evaluation of piperidinyl-substituted [1,2,4]triazolo[1,5-a]pyrimidine derivatives as potential anti-HIV-1 agents with reduced cytotoxicity. Chemical Biology & Drug Design, 97, 67, 2021.
2021-04
[8] 张涛. The development of an effective synthetic route of rilpivirine. BMC CHEMISTRY, 15, 2021.
2021-03
[9] 姜向毅. Exploiting the tolerant region I of the non-nucleoside reverse transcriptase inhibitor (NNRTI) binding pocket. Part 2: Discovery of diarylpyrimidine derivatives as potent HIV-1 NNRTIs with high Fsp(3) values and favorable drug-like properties. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 213, 2021.
2021-03
[10] 孙彦莹. Identification of novel potent HIV-1 inhibitors by exploiting the tolerant regions of the NNRTIs binding pocket. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 214, 2021.

TOTAL 27 PIECE 1/3

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