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Design, synthesis, and biological evaluation of novel 5-Alkyl-6-Adamantylmethylpyrimidin-4(3H)-ones as HIV-1 non-nucleoside reverse-transcriptase inhibitors

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Affiliation of Author(s):药学院

Journal:Chem Biol Drug Des

All the Authors:zhanpeng

First Author:liuxinyong

Indexed by:Unit Twenty Basic Research

Document Code:lw-183773

Volume:88

Issue:3

Page Number:380

Translation or Not:no

Date of Publication:2016-03-10

Pre One:Arylazolyl(azinyl)thioacetanilides: Part 19: Discovery of Novel Substituted Imidazo[4,5-b]pyridin-2-ylthioacetanilides as Potent HIV NNRTIs Via a Structure-based Bioisosterism Approach

Next One:Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approach