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Structure-based Bioisosterism Design, Synthesis and Biological Evaluation of Novel 1,2,4-Triazin-6-ylthioacetamides As Potent HIV-1 NNRTIs.

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Affiliation of Author(s):药学院

Journal:Bioorg. Med. Chem. Lett.

All the Authors:liuxinyong

First Author:展鹏

Indexed by:Unit Twenty Basic Research

Document Code:lw-135744

Volume:22

Issue:23

Page Number:7155

Translation or Not:no

Date of Publication:2012-10-15

Pre One:Discovery of Novel 2-(3-(2-Chlorophenyl) pyrazin-2-ylthio)-N-arylacetamides As Potent HIV-1 Inhibitors Using a Structure-Based Bioisosterism Approach.

Next One:Arylazolyl(azinyl)thioacetanilide. Part 9: Synthesis and Biological Investigation of Thiazolylthioacetamides Derivatives as a Novel Class of Potential Antiviral Agents.