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黄伯世.
Structure-Based Design and Discovery of Pyridyl-Bearing Fused Bicyclic HIV-1 Inhibitors: Synthesis, Biological Characterization, and Molecular Modeling Studies.
Journal of Medicianal Chemistry,
64,
13604-13621,
2023.
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黄伯世.
First discovery of a potential carbonate prodrug of NNRTI drug candidate RDEA427 with submicromolar inhibitory activity against HIV-1 K103N/Y181C double mutant strain.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
28,
1348,
2023.
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Design of bivalent ligands targeting putative GPCR dimers.
Drug Discovery Today,
26,
189-199,
2022.
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Teaching an old dog new tricks: Drug discovery by repositioning natural products and their derivatives.
Drug Discovery Today,
27,
1936-1944,
2022.
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Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV-1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles.
Journal of Medicinal Chemistry,
62,
2083–2098,
2022.
